平安! 发表于 2011-11-9 19:57
: d# v6 [' x! A! |* IPazopanib (100 mg/kg/day free base equivalent) + a1 M' ?* H. F- F
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。8 S+ f2 V+ w" |7 m' Q* P
搜索了一下,原料一大堆。
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对不起!100mg/kg是用于移植瘤的,我弄错了。+ v# _6 y# X, K& b7 _
3 ~ C' t% O) u+ ^+ o; L! }5 R以下是正版说明书的推荐用量。3 [& t* A L% @4 W j& C
, z+ x4 X. [/ V2 N: G+ p2 r: ^) u--------------------- DOSAGE AND ADMINISTRATION ----------------8 C% H6 i& j/ c( O" P
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
+ i8 @ z( f# _+ d. I% r* U* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) 2 G' L3 s% w2 V% y' r7 b; H3 V! R
---------------------DOSAGE FORMS AND STRENGTHS --------------+ v. F- K4 q( ]+ u3 ]3 e
200 mg tablets. (3) - i0 I; T- k/ x0 @+ k! V
-------------------------------CONTRAINDICATIONS------------------------ |