平安! 发表于 2011-11-9 19:57
& d0 N2 @% g4 V8 oPazopanib (100 mg/kg/day free base equivalent)
7 B! W& K/ C1 o- {" Z 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。$ B+ @8 [2 Q/ b/ t, C+ T9 z
搜索了一下,原料一大堆。7 F( i2 s: }% }
. q& v4 M4 L7 o) V- N' G对不起!100mg/kg是用于移植瘤的,我弄错了。1 ?) l- L& L7 A
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以下是正版说明书的推荐用量。
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% R; x0 v8 @! o--------------------- DOSAGE AND ADMINISTRATION ----------------
5 s4 {( Y% U" g# W5 O; F* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
& S. |) B3 O" f5 z) n/ C o; U) `* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
% C" x, L5 L& E9 L: P5 N) b. e% {---------------------DOSAGE FORMS AND STRENGTHS --------------3 H+ x/ y, h1 l4 C# A
200 mg tablets. (3)
% J! B! d+ R4 i5 K* g9 n-------------------------------CONTRAINDICATIONS------------------------ |