平安! 发表于 2011-11-9 19:57 8 I1 t; ~: ~6 n' y+ }5 D/ Y/ f. M
Pazopanib (100 mg/kg/day free base equivalent)
8 `' R- g% T0 K# l. _ 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。
/ p: k. q0 p% \; n4 H3 I2 ?搜索了一下,原料一大堆。
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4 P- R! ?0 q7 e' ]- O0 |# p. P对不起!100mg/kg是用于移植瘤的,我弄错了。$ g2 A6 g5 f% C% n& I" X- A
9 W/ X+ U% R% t) B* f以下是正版说明书的推荐用量。/ k* |0 O! m9 R0 U. ~
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--------------------- DOSAGE AND ADMINISTRATION ----------------
: S9 Q) z. O% V* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
, k6 o* M) X, [0 }3 T. }* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
! l9 W9 L% n7 W3 x8 [---------------------DOSAGE FORMS AND STRENGTHS --------------
$ M# \, P. m# G) [! D( B200 mg tablets. (3)
8 E- E% a% S6 C2 c3 S- y-------------------------------CONTRAINDICATIONS------------------------ |